2014  
  1. D'Amore C., Di Leva FS., Sepe V., Renga B., Del Gaudio C., D'Auria MV., Zampella A., Fiorucci S., Limongelli V. Design, synthesis and biological evaluation of potent dual agonists of nuclear and membrane bile acid receptors. J Med Chem. 2014, 57, 937-954. doi: 10.1021/jm401873d
  2. Domínguez, HJ., Napolitano, JG., Fernández-Sánchez, MT., Cabrera-García, D., Novelli, A., Norte, M., Fernández, JJ., Hernández Daranas, A. Belizentrin, a Bioactive Macrolide from the Dinoflagellate Prorocentrum belizeanum, Org. Lett. 2014, 6, 4546-4549. DOI: 10.1021/ol502102f
  3. Domínguez, HJ., Crespín, GD., Santiago-Benítez, AJ.; Gavín, JA., Norte, M., Fernández, JJ., Hernández Daranas A. Stereochemistry of  Complex  Marine Natural Products by Quantum Mechanical Calculations of NMR Chemical  Shifts: Solvent and Conformational  Effects on Okadaic Acid. Mar. Drugs, 2014, 12, 176-192. doi:10.3390/md12010176 
  4.  Felczykowska, A., Dydecka, A., Bohdanowicz, M., Gąsior, T., Soboň, M., Kobos, J., Bloch, S., Nejman-Faleńczyk, B., Węgrzyn, G. The use of fosmid metagenomic 1 libraries in  preliminary screening for various biological activities. Microbial Cell Factories 2014, 13:105, 1-7.
  5. Gutiérrez-Cepeda, A., Hernández Daranas, A., Fernández, JJ., Norte, M., Souto, ML, Stereochemical Determination of Five-Membered Cyclic Ether Acetogenins Using a Spin-Spin Coupling Constant Approach and DFT Calculations. Mar. Drugs 2014, 12, 4031-4044. doi:10.3390/md12074031
  6. Hodnik, Ž., Peterlin Mašič, L., Tomašić, T., Smodiš, D., D'Amore, C., Fiorucci, S., Kikelj, D., Bazedoxifene scaffold-based mimetics of solomonsterols A and B as novel pregnane X receptor antagonists, J. Med. Chem. 2014, 57, 4819-4833. DOI: 10.1021/jm500351m
  7. Hodnik, Ž., Łoś, JM., Žula, A., Zidar, N., Jakopin, Ž., Łoś, M., Sollner Dolenc M., Ilaš, J., Węgrzyn, G., Peterlin Mašič, L., Kikelj, D. Inhibition of biofilm formation by conformationally constrained indole-based analogues of the marine alkaloid oroidin, Bioorg. Med. Chem. Lett. 2014, 24, 2530-2534.
  8. Imamoglu, E., Demirel, Z., Conk Dalay, M., A Response Surface Methodology Study for the Protein Production of Chlorella sp., Int. J. Adv. Chem. Engg. Biol. Sci. (IJACEBS) 2014, 1, 76-79. DOI: 10.15242/IJACEBS.C514068.
  9. Jukič, M., Kikelj, D., Anderluh, M. Isoform Selective Voltage-Gated Sodium Channel Modulators and the Therapy of Pain, Curr. Med. Chem., 2014, 21, 164-186.
  10. Kiuru, P., D'Auria, MV., Muller, CD., Tammela, P., Yli-Kauhaluoma, J., Vuorela, H. Exploring Marine Resources for Bioactive Compounds, Planta Med. 2014, 80, 1234-46.
  11. Lebbe, EK., Peigneur, S., Brullot, W., Verbiest, T., Tytgat J. Ala-7, His-10 and Arg-12 are crucial amino acids for activity of a synthetically engineered μ-conotoxin. Peptides 2014, 53, 300-306 pii: S0196-9781(13)00234-9. doi:0.1016/j.peptides.2013.07.005.
  12. Lebbe, EKM., Peigneur, S., Maiti, M., Devi, P., Ravichandran, S., Lescrinier, E., Waelken, E., D'Souza, L., Herdewijn, P., Tytgat, J. Structure-Function Elucidation of a New α-conotoxin, Lo1a, from Conus longurionis. J. Biol. Chem. 2014, 289, 9573-9583. doi: 10.1074/jbc.M114.556175
  13. Lebbe, EKM., Peigneur, S., Wijesekara, I., Tytgat, J. Conotoxins targeting nicotinic acetylcholine receptors: an overview. Mar. Drugs 2014, 12, 2970-3004. doi:10.3390/md12052970
  14. Lillsunde, K-E., Festa, C., Adel, H., De Marino, S., Lombardi, V., Tilvi, S., Nawrot, DA., Zampella, A., D'Souza, L., D'Auria, MV., Tammela, P. Bioactive cembrane derivatives from the Indian Ocean soft coral Sinularia kavarattiensis, Mar. Drugs 2014, 12, 4045-4068. doi:10.3390/md12074045
  15. Majik, MS., Rodrigues, C., Mascarenhas,S., D'Souza, L. Design and synthesis of marine natural product-based 1H-indole-2,3-dione scaffold as a new antifouling/ antibacterial agent against fouling bacteria. Bioorg. Chem. 2014, 54, 89-95. DOI: 10.1016/j.bioorg.2014.05.001
  16. Majik, MS., Parvatkar, PT., Next Generation Biofilm Inhibitors for Pseudomonas aeruginosa: Synthesis and Rational Design Approaches. Curr. Topics Med. Chem., 2014, 14, 81-109.
  17. Majik, MS., Shirodkar, D., Rodrigues, C., D'Souza, L., Tilvi, S. Evaluation of single and joint effect of metabolites isolated from marine sponges, Fasciospongia cavernosa and Axinella donnani on antimicrobial properties. Bioorg. Med. Chem. Lett. 2014, 24, 2863-2866.
  18. Majik, MS., Tilvi, S., Parvatkar PT., Recent development on the synthesis of Varitriol, an antitumour agent from marine derived fungus, Emericella variecolor. Curr. Org. Synth. 2014, 11, 268-287. DOI:10.2174/1570179410666131124134200
  19. Majik, MS., Tilvi, S., Mascarenhas, S., Kumar, V., Chatterjee, A., Banerjee,M. Construction and screening of 2-arylbenzimidazole library identifies a new antifouling and Antifungal agent. RSC Adv, 2014, 4, 28259-28264. DOI:10.1039/c4ra00860j
  20. Mencarelli, A., D'Amore, C., Renga, B., Cipriani S., Carino A., Sepe, V., Perissutti, E, D'Auria, MV., Zampella, A., Distrutti, E., Fiorucci, S. Solomonsterol A, a Marine Pregnane-X-Receptor Agonist, Attenuates Inflammation and Immune Dysfunction in a Mouse Model of Arthritis. Mar. Drugs 2014, 12, 36-53. doi:10.3390/md12010036
  21. Peigneur, S., Žula, A., Zidar N., Chan-Porter, F., Kirby, R., Madge, D., Ilaš, J., Kikelj, D. Action of Clathrodin and Analogues on Voltage-Gated Sodium Channels. Mar. Drugs 2014, 12, 2132-2143. doi:10.3390/md12042132
  22. Parvatkar, PT., Majik, MS., Microwave-assisted reductive cyclization:  An easy entry to the indoloquinolines and spiro[2H-indole-2,3'-oxindole], RSC Adv. 2014, 4, 22481-22486. DOI: 10.1039/C4RA02814G
  23. Parvatkar, PT., Kadam, HK., Tilve, SG. Intramolecular Diels-Alder reaction as a key step in tandem or sequential processes: a versatile tool for the synthesis of fused and bridged bicyclic or polycyclic compounds, Tetrahedron, 2014, 70, 2857-2888. DOI: 10.1016/j.tet.2014.02.048
  24. Schwenk, D., Nohynek, L., Rischer, H., Algae-bacteria association inferred by 16S rDNA similarity in established microalgae cultures, Microbiol Open, 2014, 3, 356-368. DOI: 10.1002/mbo3.175
  25. Sepe, V., D'Amore, C., Ummarino, R., Renga, B., D'Auria, MV., Novellino, E., Sinisi, A., Taglialatela-Scafati, O., Nakao, Y., Limongelli, V., Zampella, A., Fiorucci S. Insights on Pregnane-X-Receptor Modulation. Natural and Semisynthetic Steroids from Theonella Marine Sponges Eur. J. Med. Chem. 2014, 73, 126-134.http://dx.doi.org/10.1016/j.ejmech.2013.12.005
  26. Sepe V., Di Leva, FS., D'Amore, C., Festa, C., De Marino, S., Renga, B., D'Auria, MV., Novellino, E., Limongelli, V., D'Souza, L., Majik, M., Zampella, A., Fiorucci, S. Marine and semi-synthetic hydroxysteroids as new scaffolds for pregnane X receptor modulation, Mar. Drugs 2014, 12, 3091-3115. doi:10.3390/md12063091
  27. Singh, K.S., Majik M. S., Tilvi, S. 2014, Vibrational spectroscopy for structural characterization of bioactive compounds in Comprehensive Analytical Chemistry Vol 65, Analysis of Marine sample in search of bioactive compounds Eds. Rocha-Santos T and Duarte AC, Elsevier, 115-148.
  28. Tilvi, S., Majik MS., Singh, KS. 2014 Mass spectrometry for determination of bioactive compounds in Comprehensive Analytical Chemistry Vol 65, Analysis of Marine sample in search of bioactive compounds, Eds. Rocha-Santos T and Duarte AC, Elsevier, 193-218.
  29. Zidar N, Jakopin Z, Madge DJ, Chan F, Tytgat J, Peigneur S, Dolenc MS, Tomašić T, Ilaš J, Mašič LP, Kikelj D. Substituted 4-phenyl-2-aminoimidazoles and 4-phenyl-4,5-dihydro-2-aminoimidazoles as voltage-gated sodium channel modulators. Eur. J. Med. Chem. 2014, 74C, 23-30. doi: 10.1016/j.ejmech.2013.12.034.
  30. Zidar, N., Montalvão, S, Hodnik, Z., Nawrot DA., Žula, A., Ilaš, J., Kikelj, D., Tammela, P., Peterlin Mašič,L. Antimicrobial Activity of the Marine Alkaloids, Clathrodin and Oroidin, and Their Synthetic Analogues, Mar. Drugs 2014, 12, 940-963. doi:10.3390/md12020940
  31. Žula, A., Kikelj, D., Ilaš, J., A convenient strategy for synthesising Agelas alkaloids clathrodin, oroidin and hymenidin and their (un)saturated linker analogs, Tetrahedron Lett. 2014, 55, 3999-4001. DOI:10.1016/j.tetlet.2014.05.087
  32. Vergauwe, N., Vermeir, S., Wacker, J., Ceyssens, F., Cornaglia, M., Puers, B., Gijs, M., Lammertyn, J., Witters, D.A highly efficient extraction protocol for magnetic particles on a digital microfluidic chip.Sensors Actuators B, Chem. 2014, 196, 282-291. DOI 10.1016/j.snb.2014.01.076   

 2013  
  1. Bergeron ZL, Chun JB, Baker MR, Sandall DW, Peigneur S, Yu PY, Thapa P, Milisen JW, Tytgat J, Livett BG, Bingham JP. A 'conovenomic' analysis of the milked venom from the mollusk-hunting cone snail Conus textile-the pharmacological importance of post-translational modifications. Peptides. 2013, 49, 145-58. doi: 10.1016/j.peptides.2013.09.004. 
  1. Cassoli JS, Verano-Braga T, Oliveira JS, Montandon GG, Cologna CT, Peigneur S, Pimenta AM, Kjeldsen F, Roepstorff P, Tytgat J, de Lima ME. The proteomic profile of Stichodactyla duerdeni secretion reveals the presence of a novel O-linked glycopeptides. J. Proteomics 2013, 87, 89-102. doi: 10.1016/j.jprot.2013.05.022. 
  1. Cen-Pacheco, F., Rodríguez, J., Norte, M., Fernández, JJ., Hernández Daranas, A. Connecting Discrete Stereoclusters by Using DFT and NMR Spectroscopy: The Case of Nivariol. Chem. Eur. J. 2013, 19, 8525-8532. DOI 10.1002/chem.201204272 
  1. Chugunov AO, Koromyslova AD, Berkut AA, Peigneur S, Tytgat J, Polyansky AA, Pentkovsky VM, Vassilevski AA, Grishin EV, Efremov RG. Modular organization of α-toxins from scorpion venom mirrors domain structure of their targets, sodium channels. J. Biol. Chem. 2013, 288, 19014-27. doi: 10.1074/jbc.M112.431650. 
  1. Devi, P., Ravichandran, S., Ribeiro, M., Ciavatta M. L. Antifungal Potential of Marine Sponge Extract against Plant and Fish Pathogenic Fungi. Oceanography 2013, 1, 1-4. http://dx.doi.org/10.4172/2332-2632.1000112 
  1. Di Leva, FS., Festa, C., D'Amore, C., De Marino, S., Renga, B., D'Auria, MV., Novellino, E., Limongelli, V., Zampella, A., Fiorucci, S. Binding mechanism of the farnesoid X receptor marine antagonist suvanine reveals a strategy to forestall drug modulation on nuclear receptors. Design, synthesis, and biological evaluation of novel ligands. J. Med. Chem. 2013, 56, 4701-17. doi: 10.1021/jm400419e 
  1. Hodnik, Ž., Tihomir T., Peterlin Mašič, L., Chan, F., Kirby, RW., Madge, DJ., Kikelj, D. Novel state-dependent voltage-gated sodium channel modulators, based on marine alkaloids from Agelas sponges. Eur. J. Med. Chem. 2013, 70, 154-64. doi: 10.1016/j.ejmech.2013.07.034 
  1. Janssen KPF., Knez, K., Spasic, D., Lammertyn, J. Nucleic acids for ultra-sensitive protein detection. Sensors, 2013, 13, 1353-84. 
  1. Kaczynska, A., Los, M., Wegrzyn G. An improved method for efficient isolation and purification of genomic DNA from filamentous cyanobacteria belonging to genera Anabaena, Nodularia and Nostoc. Oceanol. Hydrobiol. Studies 2013, 42, 8-13. DOI: 10.2478/s13545-013-0058-y 
  1. Kendel, Y., Melaun, C., Kurz, A., Nicke, A., Peigneur, S., Tytgat, J., Wunder, C., Mebs, D., Kauferstein, S.. Venomous secretions from marine snails of the Terebridae family target acetylcholine receptors. Toxins (Basel). 2013, 5, 1043-50. doi: 10.3390/toxins5051043. 
  1. Lehmann, N., Rischer, H., Eibl, D. and Eibl, R. Wave-mixed and orbitally shaken single-use photobioreactors for diatom algae propagation, Chem. Ing. Tech. 2013, 85, 1-6. 
  1. Mazur-Marzec, H., Kaczkowska, MJ., Blaszczyk, A., Akcaalan, R., Spoof, L. and Meriluoto, J. Diversity of peptides produced by Nodularia spumigena from various geographical regions. Mar. Drugs 2013, 11, 1-19. doi:10.3390/md11010001 
  1. Naik, DN., Wahidullah, S. and Meena, RM., Attenuation of Pseudomonas aeruginosa virulence by marine invertebrate-derived Streptomyces sp.. Lett. Appl. Microbiol. 2013, 56, 197-207. 
  1. Orts, DJ., Moran, Y., Cologna, CT., Peigneur, S., Madio, B., Praher, D., Quinton, L., De Pauw, E., Bicudo, JE., Tytgat, J., de Freitas, JC. BcsTx3 is a founder of a novel sea anemone toxin family of potassium channel blocker. FEBS J. 2013, 280, 4839-4852. doi: 10.1111/febs.12456. 
  1. Petrel, C., Hocking, HG., Reynaud, M., Upert, G., Favreau, P., Biass, D., Paolini-Bertrand, M., Peigneur, S., Tytgat, J., Gilles, N., Hartley, O., Boelens, R., Stocklin, R., Servent, D. Identification, structural and pharmacological characterization of τ-CnVA, a conopeptide that selectively interacts with somatostatin sst3 receptor. Biochem. Pharmacol. 2013, 85, 1663-71. doi: 10.1016/j.bcp.2013.03.019. 
  1. Rodríguez, AA., Salceda, E., Garateix, AG., Zaharenko, AJ., Peigneur, S., López, O., Pons, T., Richardson, M., Díaz, M., Hernández, Y., Ständker, L., Tytgat, J., Soto, E. A novel sea anemone peptide that inhibits acid-sensing ion channels. Peptides. 2013 pii: S0196-9781 (13) 00220-9. doi: 10.1016/j.peptides.2013.06.003.
  1. Saab, L., Peluso, J., Muller, CD., Ubeaud-Sequier. G. Implication of hepatic transporters (MDR1 and MRP2) in inflammation-associated idiosyncratic drug-induced hepatotoxicity investigated by microvolumecytometry. Cytometry A, 2013, 83A, 403-408. 
  1. Schwenk, D., Seppälä, J., Spilling, K., Virkki, A., Tamminen, T., Oksman-Caldentey, K.-M., Rischer, H., Lipid content in 19 brackish and marine microalgae: influence by growth phase, salinity and temperature. Aquatic Ecol, 2013, 47, 415-424. DOI 10.1007/s10452-013-9454-z 
  1. Spasic, D., Janssen, KP., Toffalini, F., Tran, DT., Leirs, K., Decrop, D., Lammertyn, J. Integrating aptamers into micro- and nanobiosystems for diagnostics, Transducers & Eurosensors 2013, Barcelona, Spain, 16-20 June 2013, 2775-2778, Proceedings, 
  1. Tomašić, T., Hartzoulakis, B., Zidar, N., Chan, F., Kirby, RW., Madge, DJ., Peigneur, S., Tytgat, J., Kikelj, D. Ligand- and structure-based virtual screening for clathrodin-derived human voltage-gated sodium channel modulators. J. Chem. Inf. Model. 2013, 53, 3223-32. doi: 10.1021/ci400505e. 
  1. Wang, Y., Rischer, H., Eriksen, NT., Wiebe, MG. Mixotrophic continuous flow cultivation of Chlorella protothecoides for lipids. Bioresource Techn. 2013, 144, 608-614., DOI: 10.1016/j.biortech.2013.07.027 
  1. Žula, A., Kikelj, D., Ilaš, J. 2-Aminoimidazoles in medicinal chemistry. Mini Rev. Med. Chem. 2013, 13, 1921-1943.
2012 

  1. Cen Pacheco, F., Villa-Pulgarin, JA., Mollinedo, F., Norte Martín, M., Fernández JJ., Hernández Daranas, A. Saiyacenols A and B, the Key to Solve the Controversy about the Configuration of Aplysiols. Tetrahedron 2012, 68, 7275-7279. 
  1. Janssen, KPF., Knez, K., Vanysacker, L., Schrooten, J., Spasic, D., Lammertyn, J. Enabling fiber optic serotyping of pathogenic bacteria through improved anti-fouling functional surfaces. Nanotechnology 2012, 23, 235503 (7pp) 
  1. Janssen, KPF., Knez, K., Spasic, D., Schrooten, J., Lammertyn, J. Multiplexed protein detection using an affinity aptamer amplification assay. Anal. Bioanal. Chem. 2012, 404, 2073-2081. 
  1. Renga, B., Mencarelli, A., D'Amore, C., Cipriani, S., D'Auria, MV., Sepe, V., Chini, MG., Maria Monti, MC., Bifulco, G., Zampella, A., Fiorucci, S. Discovery of theonellasterol a marine sponge sterol as a highly selective FXR antagonist that protects against liver injury in cholestasis, PLoS ONE 2012, 7, e30443. doi:10.1371/journal.pone.0030443 
  1. Sepe, V., Ummarino, R., D'Auria, MV., Lauro, G., Bifulco, G., D'Amore, C., Renga, B., Fiorucci, S., Zampella, A. Modification in the side chain of solomonsterol A: discovery of cholestan disulfate as a potent pregnane-X-receptor agonist. Org. Biomol. Chem., 2012, 10, 6350-6362. 
  1. Sepe, V., Ummarino, R., D'Auria, MV., Taglialatela-Scafati,O., De Marino, S., D'Amore, C., Renga, B., Chini, MG., Bifulco, G., Nakao, Y., Fusetani, N., Fiorucci, S., Zampella, A. Preliminary Structure-Activity Relationship on Theonellasterol,a New Chemotype of FXR Antagonist, from the Marine Sponge Theonella swinhoei. Mar Drugs 2012, 10, 2448-2466. doi:10.3390/md10112448 
  1. Sepe, V., Ummarino, R., D'Auria, MV., Renga, B., Fiorucci, S., Zampella, A. The First Total Synthesis of Solomonsterol B, a Marine Pregnane X Receptor Agonist, Eur. J. Org. Chem., 2012, 5187-5194. DOI:10.1002/ejoc.201200619
  2. Tilvi, S. D'Souza, L. Identifying the related compounds using electrospray ionization tandem mass spectrometry: Bromotyrosine alkaloids from marine sponge Psammaplysilla purpurea, Eur J Mass Spectrom 2012, 18, 333-43.  
  1. Vilches-Romero, TS., Norte, M., Hernández Daranas, A. Fernández, JJ. Biosynthetic studies on water-soluble derivative 5c (DTX5c). Mar. Drugs 2012, 10, 2234-2245
  2011  
  1. Cen Pacheco, F., Villa-Pulgarin, JA., Mollinedo, F., Norte Martín, M., Fernández JJ., Hernández Daranas, A. New Polyether Triterpenes from Laurencia viridis and their Biological Evaluation Mar. Drugs 2011, 9, 2220-2235. doi:10.3390/md9112220 
  1. Janssen, KPF., Knez, K., Pollet, J., Roberts, SJ., Schrooten, J., Lammertyn, J. Assay design considerations for use of affinity aptamer amplification in ultra-sensitive protein assays using capillary electrophoresis. Anal. Methods 2011, 3, 2156-2159. 
  1. Kiuru, P. and Yli-Kauhaluoma, J. 2011 Pyridine and Its Derivatives in Heterocycles, in Natural Product Synthesis. Majumdar, K. C. and Chattopadhyay, C. K. (eds.). Weinheim, Wiley-VCH, p. 267-297. 
  1. Sepe, V., Ummarino, R., D'Auria, MV., Mencarelli, A., D'Amore, C., Renga, B., Zampella, A., Fiorucci, S. Total Synthesis and Pharmacological Characterization of Solomonsterol A, a Potent Marine Pregnane-X-Receptor Agonist Endowed with Anti-Inflammatory Activity, J. Med. Chem. 2011, 54, 4590-4599.